目前用于口服降糖的药物包括磺脲类药物、双胍类药物、α-糖苷酶抑制剂、噻唑烷二酮类药物和DPP-4抑制剂。其中属于二肽基肽酶-4(DPP-4)抑制剂的西格列汀,主要适用于II 型糖尿病,可单独应用,也可与其他药物进行组合治疗。其优点是有效降低因低血糖及体重增加引起不良反应的发生率。
百灵威供应多种糖尿病药物关键原料及中间体、离子对试剂、顶空试剂、LC-MS试剂等产品,助力企业研发与生产。
| 品名 | CAS | 货号 |
|---|---|---|
| Methyl 3-amino-4-(2,4,5-trifluorophenyl)butanoate, 95% 3-氨基-4-(2,4,5-三氟苯基)丁酸甲酯 , 95% | 1253055-92-3 | 2110929 |
| Methyl 3-oxo-4-(2,4,5-trifluorophenyl)butanoate, 98% 3-氧代-4-(2,4,5-三氟苯基)丁酸甲酯 , 98% | 769195-26-8 | 1415192 |
| Chloro(1,5-cyclooctadiene)rhodium(I) dimer, 98% (1,5-环辛二烯)氯化铑(I)二聚体 , 98% | 12092-47-6 | 190993 |
| Dichloro(cycloocta-1,5-diene)ruthenium(II), 97% 二氯(环辛基-1,5-二烯)钌(II) , 97% | 50982-12-2 | 104033 |
| N,N'-Dicyclohexylcarbodiimide, 99% N,N'-二环己基碳二亚胺 , 99% | 538-75-0 | 275928 |
| N,N-Diisopropylethylamine, 99%, for synthesis N,N-二异丙基乙胺 , 99% , 用于合成 | 7087-68-5 | 901887 |
| N,N-Dimethylacetamide, 99%, for spectroscopy N,N-二甲基乙酰胺 , 99% , 用于光谱分析 | 127-19-5 | 928320 |
| 4-Dimethylaminopyridine, 99%, for synthesis 4-二甲氨基吡啶 , 99% , 用于合成 | 1122-58-3 | 212279 |
| Pivaloyl chloride, 99% 新戊酰氯 , 99% | 3282-30-2 | 200556 |
| 2,4,5-Trifluorophenylacetic acid, 99% 2,4,5-三氟苯乙酸 | 209995-38-0 | 337797 |
| 品名 | CAS | 货号 |
|---|---|---|
| 2,4,5-Trifluorobenzaldehyde, 97% 2,4,5-三氟苯甲醛 , 97% | 165047-24-5 | 227272 |
| N-Acetyl Sitagliptin N-乙酰基西他列汀 | 1379666-94-0 | A187815 |
| (S)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic acid hydrochloride (S)-3-氨基-4-(2,4,5-三氟苯基)丁酸盐酸盐 | 1217809-78-3 | 243378 |
| Methyl 3-oxo-4-(2,4,5-trifluorophenyl)butanoate, 98% 3-氧代-4-(2,4,5-三氟苯基)丁酸甲酯 , 98% | 769195-26-8 | 1415192 |
| Sitagliptin EP Impurity A Phosphate 磷酸西他列汀杂质A | 823817-58-9 | R40150 |
| (R)-10-(2,4,5-trifluorobenzyl)-3-(trifluoromethyl)-6,7,10,11-tetrahydro-[1,2,4]triazolo[3,4-c][1,4,7]triazecine-8,12(5H,9H)-dione 西格列汀十元环制剂杂质 | 2088771-61-1 | S493150 |